Discovery of highly selective CRAF inhibitors, 3-carboxamido-2H-indazole-6-arylamide: In silico FBLD design, synthesis and evaluation

Synthesis of stereochemically diverse cyclic analogs of tubulysins

Discovery of 4-arylamido 3-methyl isoxazole derivatives as novel FMS kinase inhibitors

De Novo Design and Synthesis of a y-Turn Peptidomimetic Scaffold and Its Application as JNK3 Allosteric Ligand

Click approach to the discovery of 1,2,3-triazolylsalicylamides as potent Aurora kinase inhibitors

Design, synthesis and biological evaluation of benzyl 2-(1H-imidazole-1-yl)pyrimidine analogues as selective and potent Raf inhibitors

Syntheses and biological evaluation of 1-heteroaryl-2aryl-1H-benzimidazole derivatives as c-Jun N-terminal kinase inhibitors with neuroprotective effects

Synthesis and biological evaluation of 1-(6-methylpyridin-2-yl)-5-(quinoxalin-6-yl)-1,2,3-triazoles as transforming growth factor-beta type 1 receptor Idnase inhibitors

3D-QSAR studies of 1,2-diaryl-1H-benzimidazole derivatives as JNK3 inhibitors with protective effects in neuronal cells

In silico binding free energy predictability with p-p interaction energy-augmented scoring function: Benzimidazole Raf inhibitors as a case study